【中文品名】盐酸奈替康唑 【药效类别】抗真菌药>咪康唑类 【通用药名】NETICONAZOLE HYDROCHLORIDE 【中文别名】奈康唑、萘特康唑 【别 名】Atolant, Meticonazole, Neural, SS-717 【化学名称】 1H-Imidazole, 1-[(1E)-2-(methylthio)-1-[2-(pentyloxy)phenyl]ethenyl]-, monohydrochloride 【CA登记号】[130773-02-3] 【结 构 式】
【分 子 式】CHNOPS· 【分 子 量】 【收录药典】 【开发单位】SSP 【首次上市】1993年,日本 【性 状】 【用 途】局部抗真菌药,对毛癣菌和念珠菌属有效,并可望一日1次应用有效。 【药理药动】 本品有抑制真菌发育作用,在0.08μg/ml~5μg/ml浓度培养白色念珠菌时,引起麦解甾醇的合成抑制。在20μg/ml以上浓度时可引起细胞内K+和磷酸根离子的释放。对须发癣菌,可引起菌体尖端部膨大,细胞壁肥厚,细胞内细胞器断裂、变形等。 对酵母类真菌、皮肤丝状菌、花斑糠疹菌、黑色真菌及其它丝状菌显示具有与CTZ(克霉唑)、BFZ(必佛那唑)同样的或更好的抗真菌作用。而且,对临床新分离的菌株也同样有效。根据对本品最低抑菌浓度(MIC)和最低杀菌浓度(MBC)测定,显示对念珠菌属有抑菌作用和对皮肤丝状菌具有杀菌作用。抗真菌作用在 pH中性区更强,抗真菌作用随着接种菌数增多及培养天增加而降低。 【适 应 症】 本品适用于下列皮肤真菌病: 1.白癣足白癣、体白癣及股白癣。 2.皮肤念珠菌病指趾间糜烂、夹擦烂。 3.花斑糠疹。 【用法用量】 以1%的软膏或搽剂每天1次涂布于患部。 [制剂与规格]软膏剂:每克中含本品10mg。液体搽剂:每毫升中含本品10mg。 【不良反应】 有时局部可有刺激感、皮肤炎症、发红、红斑、龟裂、瘙痒、湿疹和脱屑增多。 【禁忌症】 对本品成分过敏者或有过敏史者禁用。 若有明显糜烂,不宜使用。 --------------------------------------------------------------- 原产地英文商品名: Atolant solution 1% 10mls/vial 20vials/box 原产地英文药品名: Neticonazole hydrochloride 中文参考商品译名: Atolant solution 1% 10毫升/支 20支/盒 中文参考药品译名: Neticonazole hydrochloride 生产厂家中文参考译名: Hisamitsu 生产厂家英文名: Hisamitsu --------------------------------------------------------------- 原产地英文商品名: Atolant cream 1% 10g/piece 20pieces/box 原产地英文药品名: Neticonazole hydrochloride 中文参考商品译名: Atolant cream 1% 10克/支 20支/盒 中文参考药品译名: Neticonazole hydrochloride 生产厂家中文参考译名: Hisamitsu 生产厂家英文名: Hisamitsu --------------------------------------------------------------- 原产地英文商品名: Atolant ointment 1% 10g/piece 20pieces/box 原产地英文药品名: Neticonazole hydrochloride 中文参考商品译名: Atolant ointment 1% 10克/支 20支/盒 中文参考药品译名: Neticonazole hydrochloride 生产厂家中文参考译名: Mitsubishi Tanabe 制药公司 生产厂家英文名: Mitsubishi Tanabe Pharma Corporation ---------------------------------------------------------------
Brand Name:Atolant Solution 1%
Nonproprietary (Generic) Name:Neticonazole hydrochloride Dosage Form:solution
THIS MEDICINE WORKS FOR Atolant stops the growth of/or kills fungus ( such as trichophyton or candida ) which are the main cause of a skin infection such as athlete's foot or candidiasis. BEFORE USING THIS MEDICINE Tell your Doctor: - If you ever had unusual or allergic reaction to any medicines. - Patients with severe inflammation of skin. - If you are using any other prescription or nonprescription (OTC) medicines. Pregnancy/Breast-feeding Make sure your doctor knows if you are already pregnant or are breast-feeding. HOW SHOULD THIS MEDICINE BE USED? ・Follow your doctor's instructions. Wash your hands first, then gently rub the medication in the affected and surrounding area. Use once a day. ・Keep Atolant away from eyes. In case Atolant gets in your eyes, wash with water. Consult with your eye doctor ( ophthalmologic surgeon ) if needed. ・If you are ordered to use this medicine on regular schedule and you missed a dose, apply as soon as possible. ・If you put too much Atolant, wipe off with a tissue paper. Do not reuse the wiped off solution or tissue. ・Do not stop your medication without the instructions of your doctor. SIDE EFFECT(s) OF THIS MEDICINE A medicine may cause some unwanted effects. Stop taking your medicine and check with your doctor immediately if any of the following side effects occur: Other side effects not listed above may also occur in some patients. If you notice any other effects, check with your doctor: Tingling feeling, dermatitis, skin turning red, itching, exposed raw patches of tissue, scaling/cracking skin. Check with your doctor/pharmacist if anything is bothersome to you.
于2011年10月31日更新 |